Prati
Andrei Leitão
Andrei Leitão
Professor Doutor - Instituto de Química de São Carlos, Universidade de São Paulo
Potvrđena adresa e-pošte na iqsc.usp.br
Naslov
Citirano
Citirano
Godina
In vivo effects of a GPR30 antagonist
MK Dennis, R Burai, C Ramesh, WK Petrie, SN Alcon, TK Nayak, ...
Nature chemical biology 5 (6), 421-427, 2009
5442009
Câncer e agentes antineoplásicos ciclo-celular específicos e ciclo-celular não específicos que interagem com o DNA: uma introdução
VL Almeida, A Leitão, LCB Reina, CA Montanari, CL Donnici, MTP Lopes
Química nova 28, 118-129, 2005
4272005
Novel derivatives of 1, 3, 4-oxadiazoles are potent mitostatic agents featuring strong microtubule depolymerizing activity in the sea urchin embryo and cell culture assays
AS Kiselyov, MN Semenova, NB Chernyshova, A Leitao, AV Samet, ...
European journal of medicinal chemistry 45 (5), 1683-1697, 2010
892010
Molecular design, synthesis and trypanocidal activity of dipeptidyl nitriles as cruzain inhibitors
LAA Avelar, CD Camilo, S de Albuquerque, WB Fernandes, C Gonçalez, ...
PLoS Negl Trop Dis 9 (7), e0003916, 2015
722015
Molecular design, synthesis and trypanocidal activity of dipeptidyl nitriles as cruzain inhibitors
LAA Avelar, CD Camilo, S de Albuquerque, WB Fernandes, C Gonçalez, ...
PLoS neglected tropical diseases 9 (7), e0003916, 2015
722015
Exemestane's 17-hydroxylated metabolite exerts biological effects as an androgen
EA Ariazi, A Leitao, TI Oprea, B Chen, T Louis, AM Bertucci, CGN Sharma, ...
Molecular cancer therapeutics 6 (11), 2817-2827, 2007
662007
Structure–activity relationships of novel inhibitors of glyceraldehyde-3-phosphate dehydrogenase
A Leitão, AD Andricopulo, G Oliva, MT Pupo, AA de Marchi, PC Vieira, ...
Bioorganic & medicinal chemistry letters 14 (9), 2199-2204, 2004
612004
Ligand efficiency metrics considered harmful
PW Kenny, A Leitão, CA Montanari
Journal of computer-aided molecular design 28 (7), 699-710, 2014
512014
Chk1 phosphorylation of Metnase enhances DNA repair but inhibits replication fork restart
R Hromas, EA Williamson, S Fnu, YJ Lee, SJ Park, BD Beck, JS You, ...
Oncogene 31 (38), 4245-4254, 2012
402012
Small molecule inhibitors of hantavirus infection
PR Hall, A Leitão, C Ye, K Kilpatrick, B Hjelle, TI Oprea, RS Larson
Bioorganic & medicinal chemistry letters 20 (23), 7085-7091, 2010
402010
Targeting the Transposase Domain of the DNA Repair Component Metnase to Enhance ChemotherapyTherapeutically Targeting Transposase Domains
EA Williamson, L Damiani, A Leitao, C Hu, H Hathaway, T Oprea, L Sklar, ...
Cancer research 72 (23), 6200-6208, 2012
382012
Detection of intracellular granularity induction in prostate cancer cell lines by small molecules using the HyperCyt® high-throughput flow cytometry system
MK Haynes, JJ Strouse, A Waller, A Leitao, RF Curpan, C Bologa, ...
Journal of biomolecular screening 14 (6), 596-609, 2009
372009
Can Cysteine Protease Cross-Class Inhibitors Achieve Selectivity?
L Cianni, CW Feldmann, E Gilberg, M Gütschow, L Juliano, A Leitão, ...
Journal of medicinal chemistry 62 (23), 10497-10525, 2019
342019
Experimental study and computational modelling of cruzain cysteine protease inhibition by dipeptidyl nitriles
AM Dos Santos, L Cianni, D De Vita, F Rosini, A Leitão, CA Laughton, ...
Physical Chemistry Chemical Physics 20 (37), 24317-24328, 2018
322018
Anti-trypanosomal activity of non-peptidic nitrile-based cysteine protease inhibitors
ACB Burtoloso, S de Albuquerque, M Furber, JC Gomes, C Gonçalez, ...
PLOS Neglected Tropical Diseases 11 (2), e0005343, 2017
302017
A comparative study of warheads for design of cysteine protease inhibitors
DG Silva, JFR Ribeiro, D De Vita, L Cianni, CH Franco, LH Freitas-Junior, ...
Bioorganic & Medicinal Chemistry Letters, 2017
292017
Cancer and cell cicle-specific and cell cicle nonspecific anticancer DNA-interactive agents: an introduction
VL Almeida, A Leitão, LCB Reina, CA Montanari, CL Donnici, MTP Lopes
Quimica nova 28, 118-129, 2005
292005
Cancer and cell cicle-specific and cell cicle nonspecific anticancer DNA-interactive agents: an introduction
VL Almeida, A Leitão, LCB Reina, CA Montanari, CL Donnici, MTP Lopes
Quimica nova 28, 118-129, 2005
292005
Cancer and cell cicle-specific and cell cicle nonspecific anticancer DNA-interactive agents: an introduction
VL Almeida, A Leitão, LCB Reina, CA Montanari, CL Donnici, MTP Lopes
Quimica nova 28, 118-129, 2005
292005
Characterization, solubility and biological activity of amphihilic biopolymeric Schiff bases synthesized using chitosans
HFG Barbosa, M Attjioui, A Leitão, BM Moerschbacher, ÉTG Cavalheiro
Carbohydrate polymers 220, 1-11, 2019
272019
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